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Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50074007'
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50074007(6-(3,5-dimethyl-4-isoxazolylsulfonamido)-1'-[2-(1-...)
Affinity DataKi:  0.690nMAssay Description:Ability of the compound to displace [125I]-HEAT from cloned human Alpha-1A adrenergic receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50074007(6-(3,5-dimethyl-4-isoxazolylsulfonamido)-1'-[2-(1-...)
Affinity DataKi:  10nMAssay Description:Binding affinity of the compound against Alpha-1A adrenergic receptor in human prostatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Merck

Curated by ChEMBL
LigandPNGBDBM50074007(6-(3,5-dimethyl-4-isoxazolylsulfonamido)-1'-[2-(1-...)
Affinity DataKi:  10nMAssay Description:Binding affinity of the compound against Alpha-1A adrenergic receptor in rat prostatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed