Affinity DataKi: 275nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Displacement of [3H]RX821002 from human alpha2C adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at human alpha2C adrenoreceptor expressed in CHO cells assessed as extracellular acidification measured after 4 mins by cytosensor m...More data for this Ligand-Target Pair