Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM18178'
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

LigandPNGBDBM18178(4-[(1R,7S,7aR)-7-hydroxy-3-oxo-1-(trifluoromethyl)...)
Affinity DataKi:  0.900nM ΔG°:  -51.1kJ/mole EC50:  2.5nMpH: 7.4 T: 2°CAssay Description:Receptor Binding Assay (Ki)-Binding determined through direct displacement of ligand with [3H]-DHT in the MDA-453 cell line. Transactivation Assay (E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed