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Found 2 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM426784'
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426784(US10544110, Compound 5k)
Affinity DataIC50:  3.10E+3nMAssay Description:The biological activity of analogs 5-16, 18, 20, 26, JJ-450, and the resolved enantiomers JJ-450A and J-450B was determined and compared to HTS hit 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Pittsburgh

US Patent
LigandPNGBDBM426784(US10544110, Compound 5k)
Affinity DataEC50:  3.10E+3nMAssay Description:Antagonist activity at androgen receptor in human C4-2-PSA-rl cells incubated for 24 hrs in presence of androgen R1881 by dual-glo luciferase reporte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed