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Found 2 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50069075'
TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50069075((5bR,7S,9aR)-7-Methyl-4-trifluoromethyl-1,5b,6,7,8...)
Affinity DataKi:  23nMAssay Description:Binding affinity against Androgen receptor transfected into COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50069075((5bR,7S,9aR)-7-Methyl-4-trifluoromethyl-1,5b,6,7,8...)
Affinity DataEC50:  64nMAssay Description:Antagonistic activity (IC50) against human androgen receptor (hAR) in cotransfected CV-1 cellMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed