Affinity DataIC50: 37nMAssay Description:Antagonist activity at androgen receptor F877L mutant (unknown origin) expressed in PC-3 cells assessed as inhibition of transcriptional activity mea...More data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Antagonist activity at androgen receptor F877L/T877A dual mutant (unknown origin) expressed in PC-3 cells assessed as inhibition of transcriptional a...More data for this Ligand-Target Pair