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Found 1 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM9994'
TargetAromatase(Homo sapiens (Human))
Tohoku Pharmaceutical University

LigandPNGBDBM9994((2R,8R,15S)-8-hydroxy-2,15-dimethyltetracyclo[8.7....)
Affinity DataKi:  6nM ΔG°:  -48.8kJ/mole IC50:  50nMpH: 7.5 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H] Androstenedione during aromatization. After incubation, the re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed