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Found 4 Enz. Inhib. hit(s) with Target = 'BDNF/NT-3 growth factors receptor' and Ligand = 'BDBM50528539'
TargetBDNF/NT-3 growth factors receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50528539(CHEMBL4553037)
Affinity DataIC50:  37nMAssay Description:Inhibition of His-tagged human TrkB expressed in baculovirus expression system using Tyr1 peptide as substrate after 1.5 hrs by FRET-based Z-LYTE ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBDNF/NT-3 growth factors receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50528539(CHEMBL4553037)
Affinity DataKd:  22nMAssay Description:Binding affinity to TrkB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBDNF/NT-3 growth factors receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50528539(CHEMBL4553037)
Affinity DataKd:  22nMAssay Description:Binding affinity to wild type human partial length TRKB (547 to 838 residues) expressed in mammalian expression system preincubated for 1 hr measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBDNF/NT-3 growth factors receptor(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50528539(CHEMBL4553037)
Affinity DataKd:  22nMAssay Description:Binding affinity to wild type human partial length TRKB (547 to 838 residues) expressed in mammalian expression system preincubated for 1 hr measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed