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Report error Found 2 Enz. Inhib. hit(s) with Target = 'Beta-1 adrenergic receptor' and Ligand = 'BDBM50518975'
TargetBeta-1 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518975(CHEMBL4450606)
Affinity DataKi:  269nMAssay Description:Displacement of [3H]DHA from beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes measured after 90 mins by scintilla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50518975(CHEMBL4450606)
Affinity DataIC50:  2.04E+3nMAssay Description:Antagonist activity at beta1 adrenergic receptor (unknown origin) stably expressed in HEK293 cell membranes assessed as inhibition of isoproterenol-i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed