TargetBeta-2 adrenergic receptor(Rattus norvegicus)
Niigata College of Pharmacy
Curated by PDSP Ki Database
Niigata College of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 1.35E+4nMAssay Description:Ki value was determined by accumulation of c-AMP in S-49 mouse lymphoma cells (Beta2).More data for this Ligand-Target Pair
Affinity DataKd: 1.02E+4nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
Affinity DataKd: 2.04E+4nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
Affinity DataKd: 1.58E+3nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
Affinity DataKd: 4.47E+3nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
Affinity DataKd: 1.02E+4nMAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
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