Report error Found 1 Enz. Inhib. hit(s) with Target = 'Broad substrate specificity ATP-binding cassette transporter ABCG2' and Ligand = 'BDBM50569931'
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Claude Bernard University Lyon 1
Curated by ChEMBL
Claude Bernard University Lyon 1
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of human ABCG2 transfected in human HEK293 cells assessed as inhibition of mitoxantrone efflux measured after 30 mins by FACS Calibur cyto...More data for this Ligand-Target Pair