Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM193890'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM193890((R)-4-benzyl-6-(3,5-dimethylisoxazol-4-yl)-3-ethyl...)
Affinity DataIC50:  73nMAssay Description:Inhibition of BRD4 (44 to 168 aa) (unknown origin) preincubated for 15 mins followed by substrate addition measured after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed