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Found 4 Enz. Inhib. hit(s) with Target = 'Corticotropin-releasing factor receptor 1' and Ligand = 'BDBM50148889'
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50148889(CHEMBL121896 | [3-(2,4-Dimethoxy-phenyl)-2,5-dimet...)
Affinity DataKi:  3.40nMAssay Description:Binding affinity to the cloned human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50148889(CHEMBL121896 | [3-(2,4-Dimethoxy-phenyl)-2,5-dimet...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of [125I]-o-CRF binding to CHO cells expressing human CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50148889(CHEMBL121896 | [3-(2,4-Dimethoxy-phenyl)-2,5-dimet...)
Affinity DataIC50:  76nMAssay Description:Inhibition of [125I]-o-CRF binding to CHO cells expressing human CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50148889(CHEMBL121896 | [3-(2,4-Dimethoxy-phenyl)-2,5-dimet...)
Affinity DataIC50:  76nMAssay Description:Antagonist activity at human CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed