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Found 2 Enz. Inhib. hit(s) with Target = 'Cystic fibrosis transmembrane conductance regulator' and Ligand = 'BDBM50108513'
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108513(CHEMBL3597853)
Affinity DataEC50:  5.30E+4nMAssay Description:Potentiator activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as increase in iodine influx measured after 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Istituto Giannina Gaslini

Curated by ChEMBL
LigandPNGBDBM50108513(CHEMBL3597853)
Affinity DataEC50:  5.30E+3nMAssay Description:Corrector activity at CFTR F508del mutant (unknown origin) expressed in human CFBE41o cells assessed as iodide influx after 24 hrs by HS-YFP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed