Affinity DataKi: 18nMAssay Description:Binding affinity against [3H]-U-86,170-labeled dopamine receptor D2 in cloned CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Compound was tested for agonistic activity against D2 receptor from cloned CHO cells, used [3H]U-86170 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:In vitro binding affinity against cloned mammalian dopamine D2 autoreceptor, expressed in CHO-K1 cells, using [3H]U-86170 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Compound was tested for antagonistic activity against D2 receptor from rat striatum, used [3H]raclopride as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity against [3H]-raclopride-labeled dopamine receptor D2 in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: >217nMAssay Description:Tested for affinity against cloned mammalian dopamine autoreceptor (DA) D2 receptors expressed in CHO-K1 cells using [3H]spiperone as raidoligandMore data for this Ligand-Target Pair