Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]spiperone from human dopamine D2 receptor at high affinity state expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Affinity for Dopamine receptor D2 in rat striatal membranes for high agonist state using [3H]-quinpiroleMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]quinpirole from high affinity agonist binding site of D2 receptor in Rattus norvegicus (rat) striatal membraneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Affinity of compound for the Dopamine receptor D2 in rat striatal membranes was determined for low antagonist state in rat striatal membranes using [...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Agonistic activity towards dopamine D2 receptor using radioligand [3H]-quinpirole in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Displacement of [3H]spiperone from low affinity antagonist binding site of D2 receptor in Rattus norvegicus (rat) striatal membraneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 95.1nMAssay Description:Antagonistic activity towards dopamine D2 receptor using radioligand [3H]-spiperone in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Displacement of [3H]spiperone from human dopamine D2 receptor at low affinity state expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 246nMAssay Description:Binding affinity towards human cloned dopamine (hD2s) receptors expressed in CHO cell membranes using [3H]-spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Wyeth-Ayerst Research Laboratory
Curated by ChEMBL
Affinity DataKi: 246nMAssay Description:Binding affinity to Homo sapiens (human) dopamine D2S receptorMore data for this Ligand-Target Pair
Affinity DataKi: 246nMAssay Description:Affinity towards human Dopamine receptor D2 expressed in CHO cells using [3H]-spiperoneMore data for this Ligand-Target Pair