Report error Found 23 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM85093'
Affinity DataKi: 448nMAssay Description:Binding affinity against human Dopamine receptor D2 using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 908nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 908nMAssay Description:Binding affinity at Dopamine receptor D2 in CHO cells by radioligand displacement.More data for this Ligand-Target Pair
Affinity DataKi: 920nMAssay Description:In vitro binding affinity was measured at the cloned human Dopamine receptor D2 using [3H]-spiroperidol as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Binding affinity to D2R (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Binding affinity towards cloned human Dopamine receptor D2 stably expressed in CHO cells was evaluated using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Ability to displace [3H]-spiperone from cloned human dopamine D2 receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Inhibition of human dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Binding affinity for dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor by PDSP assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.62E+3nMAssay Description:Displacement of [3H]N-methylspiperone from human D2L receptor expressed in HEK293T cell membrane incubated for 1 hr by MicroBeta scintillation counti...More data for this Ligand-Target Pair
Affinity DataKi: 1.62E+3nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.10E+3nMAssay Description:Binding affinity was evaluated for the displacement of [3H]spiperone against bovine Dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons
Curated by ChEMBL
Columbia University College of Physicians and Surgeons
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity to rat Dopamine receptor D2 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+4nMAssay Description:Displacement of [3H] Spiperone from human D2S receptor expressed in CHO cells by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.80E+4nMAssay Description:Displacement of [3H]spiroperidol from human cloned dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.80E+4nMAssay Description:In vitro binding affinity at human cloned dopamine receptor D2 (short) stably expressed in CHO cells by [3H]spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4.70E+4nMAssay Description:Displacement of [3H] Spiperone from human D2L receptor expressed in CHO cells by competitive radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.40E+4nMAssay Description:Displacement of [3H]SCH23390 from human cloned dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.40E+4nMAssay Description:In vitro binding affinity at human cloned dopamine receptor D2 (long) stably expressed in CHO cells by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Binding affinity to cloned human Dopamine receptor D2 expressed in A9L cells by [3H]spiperone displacement.More data for this Ligand-Target Pair