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Report error Found 8 Enz. Inhib. hit(s) with Target = 'D(3) dopamine receptor' and Ligand = 'BDBM50129433'
TargetD(3) dopamine receptor(Human)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50129433(CHEMBL71327 | N-{(E)-4-[4-(2,3-Dichloro-phenyl)-pi...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity for human dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50129433(CHEMBL71327 | N-{(E)-4-[4-(2,3-Dichloro-phenyl)-pi...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of [125I]IABN binding to human Dopamine D3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50129433(CHEMBL71327 | N-{(E)-4-[4-(2,3-Dichloro-phenyl)-pi...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity towards rat Dopamine receptor D3 in Sf9 cells expressing in recombinant baculovirus (Bv) using [125I]-IABN as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rat)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50129433(CHEMBL71327 | N-{(E)-4-[4-(2,3-Dichloro-phenyl)-pi...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of [125I]IABN binding to rat Dopamine D3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50129433(CHEMBL71327 | N-{(E)-4-[4-(2,3-Dichloro-phenyl)-pi...)
Affinity DataKi:  6.02nMAssay Description:Inhibition of [3H]YM-09151-2 binding to human Dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50129433(CHEMBL71327 | N-{(E)-4-[4-(2,3-Dichloro-phenyl)-pi...)
Affinity DataIC50:  7.70nMAssay Description:Stimulation of quinpirole stimulation of mitogenesis in human Dopamine receptor D3 transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50129433(CHEMBL71327 | N-{(E)-4-[4-(2,3-Dichloro-phenyl)-pi...)
Affinity DataIC50:  7.71nMAssay Description:Mitogenic stimulation or antagonism of 30 nM quinpirole-stimulated mitogenesis in CHO cells expressing human dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Human)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50129433(CHEMBL71327 | N-{(E)-4-[4-(2,3-Dichloro-phenyl)-pi...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity of quinpirole stimulation of mitogenesis in human dopamine D3 transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed