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Found 3 Enz. Inhib. hit(s) with Target = 'D(3) dopamine receptor' and Ligand = 'BDBM50253549'
TargetD(3) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuses

Curated by ChEMBL
LigandPNGBDBM50253549(3-(4-Chlorophenyl)-8-(1H-indol-3-ylmethyl)-8-azabi...)
Affinity DataKi:  15.5nMAssay Description:Displacement of [125I]IABN from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuses

Curated by ChEMBL
LigandPNGBDBM50253549(3-(4-Chlorophenyl)-8-(1H-indol-3-ylmethyl)-8-azabi...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuses

Curated by ChEMBL
LigandPNGBDBM50253549(3-(4-Chlorophenyl)-8-(1H-indol-3-ylmethyl)-8-azabi...)
Affinity DataIC50:  12.3nMAssay Description:Antagonist activity at dopamine D3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed