Found 8 Enz. Inhib. hit(s) with Target = 'DNA-dependent protein kinase catalytic subunit' and Ligand = 'BDBM50098126'
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of DNA dependent protein kinase isolated from HeLa cellsMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibitory activity against DNA-dependent protein kinase (DNA-PK)More data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of DNA-PKChecked by AuthorMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibitory activity against DNA-dependent protein kinase receptorMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of DNAPK after 2 hrs by radiometric phosphate incorporation assayMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of DNA-PK purified from human HeLa nuclear extractsMore data for this Ligand-Target Pair
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle
Curated by ChEMBL
University Of Newcastle
Curated by ChEMBL