Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM50514284'
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50514284(CHEMBL4483006)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of ERalpha in human MCF7:WS8 cells assessed as increase in degradation of ERalpha incubated for 24 hrs by In-Cell Western assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50514284(CHEMBL4483006)
Affinity DataIC50:  7.40nMAssay Description:Antagonist activity at ERalpha in human MCF7:WS8 cells incubated for 18 hrs by dual luciferase reporter gene assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed