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Found 2 Enz. Inhib. hit(s) with Target = 'Free fatty acid receptor 1' and Ligand = 'BDBM22528'
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM22528(3-(4-{[(4-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  97.7nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM22528(3-(4-{[(4-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  195nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed