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Found 5 Enz. Inhib. hit(s) with Target = 'Gamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2' and Ligand = 'BDBM50035527'
LigandPNGBDBM50035527(3-Methyl-9H-beta-carboline | CHEMBL344859)
Affinity DataKi:  8nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr,gly)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035527(3-Methyl-9H-beta-carboline | CHEMBL344859)
Affinity DataKi:  11nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr,gly,val)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035527(3-Methyl-9H-beta-carboline | CHEMBL344859)
Affinity DataKi:  39nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his,thr)beta2gama2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035527(3-Methyl-9H-beta-carboline | CHEMBL344859)
Affinity DataKi:  45nMAssay Description:Binding affinity for mutant rat GABA-A receptor alpha-6-(his)-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035527(3-Methyl-9H-beta-carboline | CHEMBL344859)
Affinity DataKi:  2.05E+3nMAssay Description:Binding affinity for rat GABA-A receptor alpha-6-beta-2-gamma-2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed