Found 8 Enz. Inhib. hit(s) with Target = 'Gastrin/cholecystokinin type B receptor' and Ligand = 'BDBM50024317'
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Montpellier
Curated by ChEMBL
University of Montpellier
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of non-sulfated CCK-8 from CCKB receptor (unknown origin) expressed in HEK cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Montpellier
Curated by ChEMBL
University of Montpellier
Curated by ChEMBL
Affinity DataKi: 19.5nMAssay Description:Binding affinity against cholecystokinin type B receptor on guinea pig cortex.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Montpellier
Curated by ChEMBL
University of Montpellier
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of [3H]pCCK-8 binding to Guinea pig cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Affinity to inhibit [3H]pCCK-8 specific binding on rat brain Cholecystokinin type B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Compound was tested for binding affinity against Cholecystokinin type B receptor expressed in CHO cells on the rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]-Bolton-Hunter CCK-8 to Cholecystokinin type B receptor in the mouse cer...More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Montpellier
Curated by ChEMBL
University of Montpellier
Curated by ChEMBL
Affinity DataKd: 22nMAssay Description:Binding affinity to CCKB receptor (unknown origin) expressed in HEK cells after 4 hrs by RP-LC-ICPMS analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair