Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Glucagon receptor' and Ligand = 'BDBM50075748'
TargetGlucagon receptor(Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075748(4-[5-(4-Chloro-phenyl)-3-cyclohexyl-1H-pyrrol-2-yl...)
Affinity DataIC50:  60nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the murine glucagon receptor (GGR) expressed on C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075748(4-[5-(4-Chloro-phenyl)-3-cyclohexyl-1H-pyrrol-2-yl...)
Affinity DataIC50:  100nMAssay Description:Binding affinity determined by reduction in binding of 125 I-glucagon to the human glucagon receptor expressed on CHO cells in absence of Mg+2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075748(4-[5-(4-Chloro-phenyl)-3-cyclohexyl-1H-pyrrol-2-yl...)
Affinity DataIC50: >3.00E+3nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50075748(4-[5-(4-Chloro-phenyl)-3-cyclohexyl-1H-pyrrol-2-yl...)
Affinity DataIC50: >3.00E+3nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]-glucagon to the human glucagon receptor (GGR) expressed on CH...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed