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Report error Found 3 Enz. Inhib. hit(s) with Target = 'Glucagon-like peptide 1 receptor' and Ligand = 'BDBM50202222'
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50202222(CHEMBL398714 | N-tert-butyl-6,7-dichloro-3-(methyl...)
Affinity DataIC50:  32nMAssay Description:Effect on augmentation of [125]GLP1 binding to human GLP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50202222(CHEMBL398714 | N-tert-butyl-6,7-dichloro-3-(methyl...)
Affinity DataEC50:  101nMAssay Description:Agonist activity at human GLP1 receptor expressed in BHK cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50202222(CHEMBL398714 | N-tert-butyl-6,7-dichloro-3-(methyl...)
Affinity DataEC50:  155nMAssay Description:Agonist activity at human GLP1 assessed as stimulation of cAMPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed