Affinity DataIC50: 1.17E+4nMAssay Description:Antagonist activity at human GRalpha expressed in HEK293 cells assessed as inhibition of dexamethasone-induced response after 24 hrs by luciferase re...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Antagonist activity at human glucocorticoid receptor-alpha expressed in HEK293 cells measured after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair