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Found 2 Enz. Inhib. hit(s) with Target = 'Gonadotropin-releasing hormone receptor' and Ligand = 'BDBM50209580'
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50209580(CHEMBL415659 | [Ncy(isopropyl)7]acyline)
Affinity DataIC50:  0.310nMAssay Description:Antagonist activity at human GnRHR expressed in HEK293 cells assessed as inhibition of GnRH-induced luciferase response by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50209580(CHEMBL415659 | [Ncy(isopropyl)7]acyline)
Affinity DataIC50:  2.5nMAssay Description:Antagonist activity at rat GnRHR expressed in HEK293 cells assessed as inhibition of GnRH-induced luciferase response by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed