Report error Found 3 Enz. Inhib. hit(s) with Target = 'Gonadotropin-releasing hormone receptor' and Ligand = 'BDBM50213666'
Affinity DataKi: 1.80nMAssay Description:Displacement of [125I]-Tyr5, DLeu6, NMeLeu7, Pro-N-Et-GnRH from cloned rat GnRHRMore data for this Ligand-Target Pair
Affinity DataIC50: 271nMAssay Description:Inhibition of human GnRHR expressed in RBL cells assessed as inhibition of GnRH-stimulated [3H]-inositol phosphate hydrolysisMore data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibition of GnRHR in rat pituitary cells assessed as inhibition of GnRH-stimulated LH releaseMore data for this Ligand-Target Pair