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Report error Found 2 Enz. Inhib. hit(s) with Target = 'Heat shock protein HSP 90-alpha' and Ligand = 'BDBM126081'
TargetHeat shock protein HSP 90-alpha(Human)
Taiho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM126081(US8779142, 100)
Affinity DataIC50:  98nMAssay Description:Displacement of biotin-labeled geldanamycin from His-tagged HSP90alpha NTD (unknown origin) preincubated for 2 hrs followed by biotin-labeled geldana...More data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Human)
Taiho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM126081(US8779142, 100)
Affinity DataIC50:  150nMpH: 7.5Assay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair