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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H1 receptor' and Ligand = 'BDBM50305262'
TargetHistamine H1 receptor(Homo sapiens (Human))
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50305262(8-Fluoro-2-methyl-5-phenethyl-2,3,4,5-tetrahydro-1...)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at histamine H1 receptor in human SK-N-SH cells assessed as histamine-induced maximum intracellular calcium spike at phase 1 trea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Chemical Diversity Research Institute

Curated by ChEMBL
LigandPNGBDBM50305262(8-Fluoro-2-methyl-5-phenethyl-2,3,4,5-tetrahydro-1...)
Affinity DataIC50:  131nMAssay Description:Antagonist activity at histamine H1 receptor in human SK-N-SH cells assessed as reduction of histamine-induced intracellular calcium spike at phase 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed