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Report error Found 5 Enz. Inhib. hit(s) with Target = 'Histamine H4 receptor' and Ligand = 'BDBM50133016'
TargetHistamine H4 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50133016((7-Chloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]histamine from recombinant human histamine H4 receptor in SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50133016((7-Chloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]- histamine from the recombinant human histamine H4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50133016((7-Chloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)...)
Affinity DataKi:  19.9nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50133016((7-Chloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)...)
Affinity DataKi:  1.90E+7nMAssay Description:Antagonist activity at Homo sapiens (human) histamine H4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetHistamine H4 receptor(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50133016((7-Chloro-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)...)
Affinity DataKi:  1.90E+7nMAssay Description:Antagonist activity at Homo sapiens (human) histamine H4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article