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Found 7 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase EZH2' and Ligand = 'BDBM50544756'
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50544756(CHEMBL4637350)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of EZH2 A677G mutant (unknown origin) by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50544756(CHEMBL4637350)
Affinity DataIC50:  7.30nMAssay Description:Inhibition of wild-type EZH2 (unknown origin) by AlphaLisa assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50544756(CHEMBL4637350)
Affinity DataIC50:  7.30nMAssay Description:Inhibition of EZH2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50544756(CHEMBL4637350)
Affinity DataIC50:  7.30nMAssay Description:Inhibition of wild-type EZH2 (unknown origin) by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50544756(CHEMBL4637350)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of wild type EZH2 (unknown origin) by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50544756(CHEMBL4637350)
Affinity DataIC50:  39nMAssay Description:Inhibition of EZH2 Y641F mutant (unknown origin) by AlphaLisa assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
West China Hospital

Curated by ChEMBL
LigandPNGBDBM50544756(CHEMBL4637350)
Affinity DataIC50:  39nMAssay Description:Inhibition of EZH2 Y641F mutant (unknown origin) by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed