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Found 1 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase EZH2 [Y641F]' and Ligand = 'BDBM441967'
TargetHistone-lysine N-methyltransferase EZH2 [Y641F](Homo sapiens (Human))
Tarapeutics Science

US Patent
LigandPNGBDBM441967(US10647700, Compound 21)
Affinity DataIC50:  103nMAssay Description:Enzymatic activity assay was conducted using EZH2(Y641F) TR-FRET assay KIT from Cisbio company on compounds that were shown to be active in primary s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent