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Found 3 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50017236'
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholi

Curated by ChEMBL
LigandPNGBDBM50017236((4aS,9aR)-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydr...)
Affinity DataKi:  450nMAssay Description:Displacement of [3H]U69593 from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholi

Curated by ChEMBL
LigandPNGBDBM50017236((4aS,9aR)-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydr...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]U69,593 from human recombinant kappa opioid receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017236((4aS,9aR)-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydr...)
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity for mouse opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed