Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50299565'
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299565((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U69-593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Clinical Research Institute Of Montreal

Curated by ChEMBL
LigandPNGBDBM50299565((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandPNGBDBM50299565((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataIC50:  3.75E+4nMAssay Description:Compound was evaluated for binding affinity towards Opioid receptor kappa 1 by displacing 125 I-DPDYNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed