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Found 5 Enz. Inhib. hit(s) with Target = 'Luciferin 4-monooxygenase' and Ligand = 'BDBM38943'
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM38943(2-(1,3-benzothiazol-2-yl)-1-phthalazinone | 2-(1,3...)
Affinity DataIC50:  150nMAssay Description:Inhibition of Photinus pyralis luciferase by Easy lite assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM38943(2-(1,3-benzothiazol-2-yl)-1-phthalazinone | 2-(1,3...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Photinus pyralis luciferase by PK-Light assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM38943(2-(1,3-benzothiazol-2-yl)-1-phthalazinone | 2-(1,3...)
Affinity DataIC50:  300nMAssay Description:Inhibition of Photinus pyralis luciferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM38943(2-(1,3-benzothiazol-2-yl)-1-phthalazinone | 2-(1,3...)
Affinity DataIC50:  600nMAssay Description:Inhibition of Photinus pyralis luciferase by Steady-Glo reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLuciferin 4-monooxygenase(Photinus pyralis)
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM38943(2-(1,3-benzothiazol-2-yl)-1-phthalazinone | 2-(1,3...)
Affinity DataIC50:  700nMAssay Description:Inhibition of Photinus pyralis luciferase by BrightGlo reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed