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Found 4 Enz. Inhib. hit(s) with Target = 'Lysosomal Pro-X carboxypeptidase' and Ligand = 'BDBM50338007'
TargetLysosomal Pro-X carboxypeptidase(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338007((S)-1-(2-(5,6-dichloro-1H-benzo[d]imidazol-2-yl)py...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of mouse PrCPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338007((S)-1-(2-(5,6-dichloro-1H-benzo[d]imidazol-2-yl)py...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human recombinant PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate after 30 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338007((S)-1-(2-(5,6-dichloro-1H-benzo[d]imidazol-2-yl)py...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human PrCPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal Pro-X carboxypeptidase(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50338007((S)-1-(2-(5,6-dichloro-1H-benzo[d]imidazol-2-yl)py...)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of PrCP in mouse plasma assessed as angiotensin 3 cleavageMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed