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Compile Data Set for Download or QSAR
maximum 50k data
Found
2
Enz. Inhib. hit(s) with Target = 'MAP kinase-activated protein kinase 2' and Ligand = 'BDBM50297113'
Target
MAP kinase-activated protein kinase 2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50297113
((R)-10-Methyl-3-pyridin-3-yl-9,10,11,12-tetrahydro...)
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Affinity Data
IC50: 5nM
Assay Description:
Inhibition of MK2
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
MAP kinase-activated protein kinase 2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50297113
((R)-10-Methyl-3-pyridin-3-yl-9,10,11,12-tetrahydro...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 220nM
Assay Description:
Inhibition of MK2 in human U937 cells assessed as blockade of LPS-stimulated TNFalpha production
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI