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Found 3 Enz. Inhib. hit(s) with Target = 'Mast/stem cell growth factor receptor Kit' and Ligand = 'BDBM8851'
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8851(3-(4-{4-amino-6-[(4-methylpiperazin-1-yl)methyl]th...)
Affinity DataIC50:  794nMAssay Description:Inhibition of cKITMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8851(3-(4-{4-amino-6-[(4-methylpiperazin-1-yl)methyl]th...)
Affinity DataIC50:  800nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Dalian University

Curated by ChEMBL
LigandPNGBDBM8851(3-(4-{4-amino-6-[(4-methylpiperazin-1-yl)methyl]th...)
Affinity DataIC50:  800nMAssay Description:Inhibition of c-Kit by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed