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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) with Target = 'Mast/stem cell growth factor receptor Kit [D816V]' and Ligand = 'BDBM369397'
Target
Mast/stem cell growth factor receptor Kit [D816V]
(Homo sapiens (Human))
Plexxikon
US Patent
Ligand
BDBM369397
((2R)-N-[(1S)-1-(4-chlorophenyl)ethyl]-4-[6- (1,3-d...)
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Affinity Data
Ki: 500nM
Assay Description:
The c-Kit mutant D816V inhibitors were assessed using an engineered BaF3-FL KIT D816V or BaF3-FL KIT V560G/D816V cell line. The BaF3-FL KIT D816V cel...
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Target Info
PDB
UniProtKB/SwissProt
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Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
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