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Found 2 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50184350'
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184350(CHEMBL409144 | c[Nle-Asp-D-Nal(2')-Arg-Trp-Glu]-NH...)
Affinity DataIC50:  170nMAssay Description:Inhibitory activity against hMC4R transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184350(CHEMBL409144 | c[Nle-Asp-D-Nal(2')-Arg-Trp-Glu]-NH...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity against hMC4R transfected in HEK293 cells by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed