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Found 3 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50266704'
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50266704(CHEMBL4083717)
Affinity DataKi:  15nMAssay Description:Antagonist activity at mouse MC4R expressed in HEK293 cells assessed as inhibition of NDP-MSH induced-cAMP accumulation after 2 hrs by alpha screen a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50266704(CHEMBL4083717)
Affinity DataIC50:  13nMAssay Description:Displacement of [125I]-NDP-MSH from mouse MC4R expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50266704(CHEMBL4083717)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed