Found 6 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 1' and Ligand = 'BDBM50030628'
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University
Curated by PDSP Ki Database
Emory University
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
Johnson and Johnson Pharmaceutical Research and Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University
Curated by PDSP Ki Database
Emory University
Curated by PDSP Ki Database
Affinity DataKi: 3.00E+4nMAssay Description:Agonist potency against cloned human metabotropic glutamate receptor 1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University
Curated by PDSP Ki Database
Emory University
Curated by PDSP Ki Database
Affinity DataIC50: 4.00E+4nMAssay Description:Ability to inhibit mGluR1-alpha-mediated PI (phospho inosotol) hydrolysis was determined at BHK cells at 100 Micro M ConcentrationMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Emory University
Curated by PDSP Ki Database
Emory University
Curated by PDSP Ki Database
Affinity DataIC50: 2.00E+5nMAssay Description:Compound was tested for inhibition of glutamate-evoked (10 uM) [Ca2+] mobilization in mGluR1-alpha expressed-CHO cells.More data for this Ligand-Target Pair