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Report error Found 1 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM116210'
TargetMu-type opioid receptor(Human)
Purde Pharma

US Patent
LigandPNGBDBM116210(US8637502, 44)
Affinity DataKi:  9.54E+3nM ΔG°:  -28.7kJ/molepH: 7.4 T: 25°CAssay Description:μ-Opioid Receptor Binding Assay Procedures: Radioligand dose-displacement binding assays for μ-opioid receptors used 0.2 nM[3H]-diprenorphi...More data for this Ligand-Target Pair
In DepthDetails US Patent