Found 6 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50001157' TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute of Montreal
Curated by ChEMBL
Clinical Research Institute of Montreal
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:. Binding affinity for Opioid receptor mu 1 determined by displacing [3H]-DAMGO from rat brain membrane binding sitesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity at mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute of Montreal
Curated by ChEMBL
Clinical Research Institute of Montreal
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute of Montreal
Curated by ChEMBL
Clinical Research Institute of Montreal
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in human/mouse HN9.10 cell membranes after 3 hrs by liquid scintillation counting ana...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileum assessed as induction of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
