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Found 5 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50272081'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50272081(2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50272081(2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity for rat brain P2 synaptosome Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50272081(2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50272081(2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...)
Affinity DataIC50:  2.60nMAssay Description:Agonist activity at mu opioid receptor by guinea pig ileum assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Cavia porcellus)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50272081(2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...)
Affinity DataIC50:  3.02nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum myenteric plexus longitudinal muscle assessed as inhibition of electrically-stimul...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed