Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M5' and Ligand = 'BDBM50241132'
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universita Di Firenze
Curated by ChEMBL
Universita Di Firenze
Curated by ChEMBL
Affinity DataKi: 0.209nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universita Di Firenze
Curated by ChEMBL
Universita Di Firenze
Curated by ChEMBL
Affinity DataKi: 0.209nMAssay Description:Displacement of [3H]N-methylscopolamine from human muscarinic M5 receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universita Di Firenze
Curated by ChEMBL
Universita Di Firenze
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-NMS from wild-type human muscarinic M5 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universita Di Firenze
Curated by ChEMBL
Universita Di Firenze
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Compound was evaluated for its binding affinity at human muscarinic receptor m5 by the displacement of [3H]-NMS radioligand using membranes from tran...More data for this Ligand-Target Pair