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Report error Found 3 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M5' and Ligand = 'BDBM50534550'
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50534550(CHEMBL4542697)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50534550(CHEMBL4542697)
Affinity DataIC50:  660nMAssay Description:Antagonist activity at human muscarinic M5 receptor assessed as inhibition of acetylcholine-induced calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50534550(CHEMBL4542697)
Affinity DataIC50:  661nMAssay Description:Antagonist activity at human muscarinic M5 receptor assessed as inhibition of acetylcholine-induced calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed