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Found 2 Enz. Inhib. hit(s) with Target = 'NAD-dependent protein deacetylase sirtuin-1' and Ligand = 'BDBM50017342'
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50017342(CHEMBL1588664)
Affinity DataIC50:  1.58E+6nMAssay Description:Inhibition of human recombinant SIRT1 assessed as reduction in NAD+-dependent deacetylase activity using Arg-His-Lys-Lys(epsilon-acetyl)-AMC substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
University of Genoa

Curated by ChEMBL
LigandPNGBDBM50017342(CHEMBL1588664)
Affinity DataIC50:  1.58E+6nMAssay Description:Inhibition of SIRT1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed